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货号 产品名 纯度
A882697 现货 Spiramide/螺拉米特

99%
A1000642 现货 ABT-724

ABT-724 is a potent and highly selective dopamine D4 receptor agonist with EC50s of 12.4 nM, 14.3 nM and 23.2 nM for human dopamine D4 receptor, rat D4 receptor and ferret D4 receptor.

98%
A819643 现货 GR 103691

GR 103691 is an effective and selective receptor antagonist of the dopamine D3 receptor (D3DR).

99%
A111766 现货 Dexpramipexole 2HCl/右旋普拉克索二盐酸盐

Dexpramipexole 2HCl is the HCl form of Dexpramipexole which is a non-ergoline dopamine agonist for treatment of parkinson's disease and restless leg syndrome.Dexpramipexole is an (R)-(+) optical enantiomer of pramipexole.

99%
A185949 现货 BP 897 HCl

BP897 is a partially selective dopamine D3 receptor agonist (Ki = 0.92 nM) that developed for the study of cocaine addiction.

99%
A669743 现货 Cabergoline/卡麦角林

Cabergoline, an ergot derivative, is a potent dopamine receptor agonist on D2 receptors.

99%
A764267 现货 Bromopride/溴必利

Bromopride is a dopamine antagonist with prokinetic properties, widely used as an antiemetic.

99%
A148362 现货 Trimethobenzamide HCl/盐酸三甲氧苯酰胺

Trimethobenzamide HCl is a dopamine D2 receptor antagonist and antiemetic drug.

99%
A447591 现货 PD-168077 maleate

PD 168077 maleate is an agonist of D4 dopamine receptor with Ki of 8.7 nM. It can induce synaptic translocation of CaMK II to postsynaptic sites in cultured prefrontal cortical neurons.

99%
A689993 现货 Dexpramipexole/右旋普拉克索

Dexpramipexole is a neuroprotective agent and weak non-ergoline dopamine agonist.

98%
A227135 现货 Brexpiprazole/依匹哌唑

Brexpiprazole is a partial agonist of the serotonin 5-HT1A receptor and the dopamine D2 and D3 receptors, used as an atypical antipsychotic for the treatment of schizophrenia and major depressive disorders.

99%
A156825 现货 (+)-PD 128907 HCl

(+)-PD 128,907 HCl is an agonist of D3 dopamine receptor with Ki of 2.3 nM.

99%
A428762 现货 Nomifensine maleate/诺米芬新马来酸盐

Nomifensine maleate is a selective inhibitor of dopamine uptake, used in adult attention deficit disorder.

98%
A308996 现货 Pardoprunox HCl

Pardoprunox HCl is a partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist.

99%
A305117 现货 Bromocriptine mesylate/甲磺酸溴隐亭

Bromocriptine mesylate is a potent dopamine D2/D3 receptoragonist, which binds D2 dopamine receptor with pKi of 8.05±0.2.

99%
A1380175 现货 Tavapadon

Tavapadon is an orally active and highly selective dopamine D1/D5 receptor partial agonist. It may be useful in the treatment of Parkinson's disease and Alzheimer's.

99%
A512636 现货 ABT-724 3HCl

ABT-724 3HCl is a potent and highly selective dopamine D4 receptor agonist with EC50s of 12.4 nM, 14.3 nM and 23.2 nM for human dopamine D4 receptor, rat D4 receptor and ferret D4 receptor.

99%
A666579 现货 Clebopride malate/苹果酸氯波必利

Clebopride malate, with antiemetic and prokinetic properties, is a dopamine antagonist drug used to treat gastrointestinal dysfunction.

99%
A115399 现货 Pramipexole 2HCl/盐酸普拉克索

Pramipexole 2HCl is an dopamine agonist and can inhibit multiple dopamine receptors including dopamine D2S receptor, dopamine D2L receptor, dopamine D3 receptor, and dopamine D4 receptor with respectively Ki values of 3.9, 2.2, 0.5 and 5.1 nM.

99%
A753188 现货 Talipexole

Talipexole is a dopamine agonist that has been proposed as an antiparkinsonian agent.

98%
产品名 D1 receptor D2 receptor D3 receptor D4 receptor D5 receptor DAT Dopamine receptor 其他靶点 纯度
Penfluridol +

Dopamine receptor, Ki: 1.6 μM

98%
Ansofaxine HCl ++

Dopamine receptor, IC50: 491 nM

99%
Tetrahydroberberine +

D2 receptor, pKi: 6.08

98+%
Prochlorperazine Maleate 98% (HPLC)
Olanzapine 99+%
Trifluoperazine ++++

Dopamine D2 receptor, IC50: 1.1 nM

98%
Ropinirole HCl ++

D2 receptor, Ki: 29 nM

99%
Lurasidone ++++

D2 receptor, Ki: 1 nM

98%
Levosulpiride 99+%
Pridopidine 95%
Metoclopramide 99+%
Molindone HCl 99%
Sulpiride 99+%
Perospirone ++++

D2 receptor, Ki: 1.4 nM

99%
Perospirone HCl ++++

D2 receptor, Ki: 1.4 nM

99%
Phenothiazine 98%
Pimozide +

Dopamine D1 receptor, Ki: 6600 nM

+++

Dopamine D2 receptor, Ki: 3.0 nM

++++

Dopamine D3 receptor, Ki: 0.83 nM

98%
Rotundine ++

D1 receptor, IC50: 166 nM

+

D2 receptor, IC50: 1.47 μM

+

D3 receptor, IC50: 3.25 μM

98%
Domperidone 99+%
ONC206 99%
Pimethixene maleate ++

Dopamine D1 Receptor, pKi: 6.37

+++

Dopamine D2 Receptor, pKi: 8.19

++

Dopamine D4.4 Receptor, pKi: 7.54

97%
Loxapine succinate ++

D2 receptor (Human), Ki: 62 nM

D1 receptor (human), Ki: 26 nM

++

D2 receptor (bovine), Ki: 26 nM

D2 receptor (human), Ki: 24 nM

+++

D4 receptor (human), Ki: 7.5 nM

98%
Chlorprothixene +++

D1 receptor, Ki: 18 nM

+++

D2 receptor, Ki: 2.96 nM

+++

D3 receptor, Ki: 4.56 nM

+++

D5 receptor, Ki: 9 nM

99%
SCH-23390 HCl ++++

D1 dopamine receptor, Ki: 0.2 nM

++++

D5 dopamine receptor, Ki: 0.3 nM

98%
MPP+ iodide 97%
σ1 Receptor antagonist-1 +

DAT, pKi: 5.8

97%
Benztropine mesylate ++

DAT, IC50: 118 nM

98%
Azaperone 98%
Ziprasidone HCl 98+%
Paliperidone 98%
Alizapride HCl 99+%
Amisulpride 98%
Quetiapine hemifumarate Adrenergic Receptor 98%
Clozapine N-oxide 99%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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