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货号 产品名 纯度
A1967304 现货 Enpp/Carbonic anhydrase-IN-2

99%
A1942416 现货 Enpp/Carbonic anhydrase-IN-1

99%
A184839 现货 1,3-Dimethyluracil/1,3-二甲基尿嘧啶

1,3-Dimethyluracil is a methyl derivative of uric acid, found occasionally in human urine.

99%
A1603338 现货 Girentuximab/吉妥昔单抗

99%
A1868758 现货 hCAII-IN-8

99%
A876758 现货 Ethoxzolamide/依索唑胺

Ethoxzolamide is an inhibitor of carbonic anhydrase with (Ki = 1 nM).

99%
A906540 现货 Benzolamide

99%
A407281 现货 Methyclothiazide/甲氯噻嗪

Methyclothiazide is a substituted benzothiadiazide, used to treat high blood pressure and fluid retention caused by various conditions including heart disease.

99%
A203568 现货 Sulfamide/磺酰胺

97%
A580496 现货 Polmacoxib

99%
A1228161 现货 Phenylsulfamide

95%
A554211 现货 2-Aminobenzenesulfonamide/2-氨基苯磺酰胺

2-Aminobenzenesulfonamide is a potent inhibitor of carbonic anhydrase B.

99%
A275314 现货 Mafenide HCl/盐酸磺胺米隆

Mafenide HCl is a sulfonamide that inhibits the enzyme carbonic anhydrase and is used as a topical anti-bacterial agent, especially in burn therapy.

99%
A119509 现货 Benzenesulphonamide/苯磺酰胺

Benzenesulfonamide ia an inhibitor of carbonic anhydrases.

99%
A1678235 现货 hCAI/II-IN-6

98%
A1258800 现货 CAIX Inhibitor S4

S4 is a selective inhibitor of CA IX and CA XII inhibitor. The Ki values are 2, 7, 547 and 5600 nM for CA XII, IX, II and I, respectively.

98%
A1417612 现货 EMAC10101d

EMAC10101d is a potent and selective Carbonic Anhydrase II inhibitor.

99%
A637802 现货 Sultiame/舒噻嗪

Sultiame is an inhibitor of carbonic anhydrase that used to treat epilepsy.

98%
A789278 现货 (R)-2-Amino-4-mercaptobutanoic acid/D-高半胱氨酸

98%
A436967 现货 Tioxolone/噻克索酮

Tioxolone, a metalloenzyme carbonic anhydrase I inhibitor with a Ki of 91 nM, is an anti-acne preparation.

99%
产品名 Carbonic Anhydrase Carbonic Anhydrase I Carbonic Anhydrase II Carbonic Anhydrase IV Carbonic Anhydrase IX Carbonic Anhydrase XII 其他靶点 纯度
Topiramate Calcium Channel 98%
Dichlorphenamide 98%
Mafenide Acetate 98%
Benzenesulphonamide 98%
Tioxolone +

CAI, Ki: 91 nM

98%
Dorzolamide HCl +

Carbonic anhydrase I, Ki: 6000 nM

++++

Carbonic anhydrase II, Ki: 1.9 nM

+++

Carbonic anhydrase IV, Ki: 31 nM

98%
Methazolamide ++

hCAI, Ki: 50 nM

+++

hCAII, Ki: 14 nM

++

bCAIV, Ki: 36 nM

98%
U-104 ++

CAIX, Ki: 45.1 nM

++++

CAXII, Ki: 4.5 nM

98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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