c-Kit

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c-Kit 相关产品
c-Kit 亚型比较

全部(113) Inhibitor(13)

货号		产品名	纯度
A725907	现货	Ripretinib/瑞普替尼 DCC-2618 is a pan-KIT and PDGFRA inhibitor, and has antitumor activity.	99%
A396655	现货	SKLB4771 FLT3-IN-1 is a potent and selective Flt3 inhibitor with IC50 of 10 nM and against FLT3-ITD-expressing MV4-11 cells with IC50 of 6 nM.	99%
A1280760	现货	Imatinib D4	99%
A1257150	现货	Telatinib mesylate	99%
A123381	现货	Motesanib/莫替沙尼 Motesanib is an ATP-competitive inhibitor of VEGFR1 (IC50 = 2 nM), VEGFR2 (IC50 = 3 nM), VEGFR3 (IC50 = 6 nM) and Kit.	99%
A394978	现货	O6-Benzylguanine O6-Benzylguanine is an inactivator of O6-alkylguanine DNA alkyltransferase (AGT) and can prevent the repair of DNA damage induced by chemotherapeutics. It induces apoptosis and cell death.	99%
A204345	现货	VEGFR-IN-1	98%
A1466435	现货	JI6	97%
A1461903	现货	Chiauranib	99%
A1216694	现货	c-Kit-IN-3	99%
A1554610	现货	Bezuclastinib	99%
A1942335	现货	Elenestinib	98%
A2417323	现货	Labuxtinib	99%
A1371593	现货	KG5	99%
A1550120	现货	M4205	99%
A1193899	现货	PD180970	99%
A172367	现货	Avapritinib BLU-285 is a potent KIT receptor and PDGFRα dual inhibitor with IC50 of 0.27 and 0.24 nM for KIT (D816V) and PDGFRα (D842V) respectively, developed as a highly targeted therapy for SM.	99%
A422593	现货	Multi-kinase inhibitor 1	99%
A314800	现货	Sitravatinib Sitravatinib is an inhibitor of receptor tyrosine kinase (RTK) involved in driving sarcoma cell growth, is developed for the treatment of cancer.	99%
A1152213	现货	Filanesib HCl	99%

产品名	c-Kit ↓ ↑	其他靶点	纯度
Tyrphostin AG1296	+ c-Kit (Swiss 3T3), IC50: 1.8 μM	PDGFR	99%+
Masitinib	+ Kit, IC50: 200 nM		99%+
Motesanib Diphosphate	+++ Kit, IC50: 8 nM		99% (HPLC)
Ki8751	++ c-Kit, IC50: 40 nM		99%
Tivozanib	++ c-Kit, IC50: 78 nM		99%+
Pazopanib	+ c-Kit, IC50: 140 nM		99%
Sitravatinib	+++ Kit, IC50: 6 nM		99%+
Pexidartinib	+++ Kit, IC50: 10 nM		99%+
Lactate	++++ c-Kit, IC50: 2 nM	FLT3	85%
Amuvatinib	+++ c-Kit (D816H), IC50: 10 nM		99%+
Imatinib Mesylate	+ c-Kit, IC50: 100 nM	PDGFR	99%
AZD2932	+++ c-Kit, IC50: 9 nM		99%
Axitinib	++++ Kit, IC50: 1.7 nM		98%
Dovitinib	++++ c-Kit, IC50: 2 nM	FLT3	99%+
Sunitinib	✔	FLT3	98%
OSI-930	+ Kit, IC50: 80 nM		99%+
Telatinib	++++ c-Kit, IC50: 1 nM		99%+
Dasatinib monohydrate	++ c-Kit (wt), IC50: 79 nM c-Kit (D816V), IC50: 37 nM	Src	98%
Dasatinib	++ c-Kit (D816V), IC50: 37 nM c-Kit (wt), IC50: 79 nM	Src	98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。

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