ZD 7155 hydrochloride is selective competitive antagonist of the angiotensin II type 1 (AT1) receptor.

Angiotensin II (3-8), human is an agonist of angiotensin AT1 receptor. Its activation is relatively weak.

AVE 0991 is a nonpeptide Ang-(1-7) receptor Mas agonist.

trans-Tranilast is an antiallergic drug, used to treat bronchial asthma, allergic rhinitis and atopic dermatitis.

Azilsartan is an orally available angiotensin II type 1 (AT1) receptor antagonist with IC50 value of 2.6 nM.

AHU-377 and valsartan can compose LCZ696 in a 1:1 molar ratio. It also works as an inhibitor of neprilysin with IC50 value of 5 nM.

Tranilast can antagonize angiotensin II and also work as an antiallergic agent. It showed inhibitory effect for NLRP3 inflammasome but not for NLRC4 or AIM2 inflammasome. Tranilast impaired the endogenous NLRP3-ASC interaction but did not affect the NLRP3-NEK7 interaction, raising the possibility that it targets NLRP3 directly.

SNOG is a NO carrier. It relaxed smooth muscle and inhibited platelet aggregation.

PD123319 Ditrifluoroacetate is a potent, selective and non-peptide angiotensin AT2 receptor antagonist.

Azilsartan Medoxomil is an orally available angiotensin II type 1 (AT1) receptor antagonist with IC50 value of 2.6 nM.

EMA401, a highly selective AT2R antagonist, inhibition of augmented AngII/AT2R induced p38 and p42/p44 MAPK activation, and hence inhibition of DRG neuron hyperexcitability and sprouting of DRG neurons.

A 779 is a specific antagonist of G-protein coupled receptor (Mas receptor), which is an Ang1-7 receptor.

Olmesartan is an antagonist of angiotensin II receptor, working as an antihypertensive agent.

EXP 3174 is a selective and noncompetitive antagonist of AT1 receptor with IC50 of 37 nM.